Top Grade Tianeptine Sodium Salt CAS NO.30123-17-2
Product Description
Tianeptine is a drug mainly used to treat major depressive disorder, although it can also be used to treat asthma or irritable bowel syndrome. Chemically, it is a tricyclic antidepressant (TCA), but it has different pharmacological properties than typical TCAs because recent studies have shown that tianeptine works by indirectly altering glutamate receptor activity (i.e. AMPA receptors and NMDA receptors) and the release of BDNF produce antidepressant effects, which in turn affect neuroplasticity.
| Product name | Tianeptine Sodium |
| CAS No. | 30123-17-2 (54317-11-2) |
| EINECS | 250-059-3 |
| Molecular formula | C21H25ClN2NaO4S |
| Molecular weight | 459.9414 |
| Appearance | Off- white to white powder |
| Solubility | DMSO: ≥20 mg/mL |
| Assay | ≥99% (HPLC) |
| Packing | 25Kg/drum |
Function
1) Tianeptine Sodium Improves Depressive Symptoms.
2) Tianeptine Sodium Lessens Anxiety, Stress, and PTSD and Symptoms From Stress.
3) Tianeptine Sodium Benefits Memory and Learning.
4) Tianeptine Sodium is an Anti-inflammatory.
5) Tianeptine Sodium decreases pain.
6) Tianeptine Sodium Helps Treat Irritable bowel Syndrome.
7) Tianeptine Sodium Reduces Asthma.
Applictaion
Tianeptine sodium salt is a salt of Tianeptine. Tianeptine, a tricyclic compound, is a selective facilitator of 5-HT (serotonin; sc-201146) uptake in vitro and in vivo. Additionally, Tianeptine is reported to act as a selective inhibitor of dopamine uptake . Tianeptine does not have a noted effect on monoamine uptake. In a study utilizing purified synaptosomes from rat brain, Tianeptine was reported to enhance serotonin uptake in selective brain regions. Purified synaptosomes were obtained from rats and incubated with tritium-labeled 5-HT and Tianeptine in vitro . The synaptosomes were then analyzed for uptake and release of 5-HT via a liquid scintillation.
Tianeptine is antidepressant. The animal has: the hippocampus pyramidal cells increased spontaneous activity, and accelerating its function was inhibited after recovery; increase in cortical and hippocampal neurons at sites of 5- serotonin reuptake. Tianeptine without following adverse effects: sleep and alertness; cardiovascular system; cholinergic system ( without anticholinergic symptoms ); drug craving.
