100% Genuine Best Quality Nootropics Tianeptine Sodium Salt 99% CAS 30123-17-2 Powder
Product Description
| Product Name | Tianeptine Sodium | Other Name | Tianeptine Sodium Salt |
| Cas No. | 30123-17-2 | MF | C21H24CLN2NAO4S |
| Einecs | 250-059-3 | Appearance | White Powder |
| Purity | 99% Min | Package | 1kg/Aluminum foil bag; 25kg/drum |
Introduction of Tianeptine sodium salt
Tianeptine sodium salt is a salt of Tianeptine. Tianeptine, a tricyclic compound, is aselective facilitator of 5-HT (serotonin; sc-201146) uptake in vitro and in vivo. Additionally,Tianeptine is reported to act as a selective inhibitor of dopamine uptake . Tianeptine doesnot have a noted effect on monoamine uptake. In study utilizing purified synaptosomesfrom rat brain, Tianeptine was reported to enhance serotonin uptake in selective brainregions. Purified synaptosomes were obtained from rats and incubated with tritium-labeled 5-HT and Tianeptine in vitro . The synaptosomes were then analyzed for uptake and releaseof 5-HT via a liquid scintillation.
Application&Function of Tianeptine sodium salt
Tianeptine has antidepressant and anxiolytic (anti-anxiety) properties with a relative lack of sedative, anticholinergic and cardiovascular adverse effects, thus suggesting it is particularly suitable for use in the elderly and in those following alcohol withdrawal; such persons can be more sensitive to the adverse effects of psychotropic drugs. Recent results indicate possible anticonvulsant (anti-seizure) and analgesic (painkilling) activity of tianeptine via immediate or downstream modulation of adenosine A1 receptors (as the effects could be experimentally blocked by antagonists of this receptor).
